• Issue

    Journal of Heterocyclic Chemistry: Volume 55, Issue 10

    2189-2440
    October 2018
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Issue Information

  • Pages: 2189-2195
  • First Published: 10 October 2018

Reviews

An Update of the Use of Thiocarbohydrazides and Thiosemicarbazides in the Preparation of Heterocycles and Their Biological Importance

Ashraf A. Aly,  Alaa A. Hassan,  El-Shaimaa S. M. AbdEl-latief, 
  • Pages: 2196-2223
  • First Published: 06 September 2018
An Update of the Use of Thiocarbohydrazides and Thiosemicarbazides in the Preparation of Heterocycles and Their Biological Importance

Recent Progress on Nicotinonitrile Scaffold-based Anticancer, Antitumor, and Antimicrobial Agents: A Literature Review

Moustafa A. Gouda,  Ehab Attia,  Mohamed H. Helal,  Mohammed A. Salem, 
  • Pages: 2224-2250
  • First Published: 31 August 2018
Recent Progress on Nicotinonitrile Scaffold-based Anticancer, Antitumor, and Antimicrobial Agents: A Literature Review

Articles

Synthesis and Antimicrobial Activity of Some Novel bis Polyfunctional Pyridine, Pyran, and Thiazole Derivatives

Elsherbiny H. El-Sayed,  Ahmed A. Fadda, 
  • Pages: 2251-2260
  • First Published: 13 August 2018
Synthesis and Antimicrobial Activity of Some Novel bis Polyfunctional Pyridine, Pyran, and Thiazole Derivatives

Design, Synthesis, Antifungal and Antibacterial Activities of N-phenyl and N-pyridinyl-5-(trifluoromethyl)-pyrazole-4-carboxamide Derivatives

Wenqing Yang,  Xiang Zhou,  Zhibing Wu, 
  • Pages: 2261-2269
  • First Published: 13 August 2018
Design, Synthesis, Antifungal and Antibacterial Activities of N-phenyl and N-pyridinyl-5-(trifluoromethyl)-pyrazole-4-carboxamide Derivatives

Three-component Strategy for Synthesis of Dihydropyrido[2,3-d]pyrimidine and Spirooxindole Derivatives

Ting Sun,  Hongdie Li,  Zhaoqi Wu,  Chunmei Li,  Xiaorong Ren,  Furen Zhang, 
  • Pages: 2270-2276
  • First Published: 17 August 2018
Three-component Strategy for Synthesis of Dihydropyrido[2,3-d]pyrimidine and Spirooxindole Derivatives

A Highly Efficient Catalyst for the Suzuki-Miyaura Cross-Coupling Reaction of 5-(5-chloropyridin-3-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one

Bhaskaran Savitha,  Eeda Koti Reddy,  D. Parthasarathi,  Rajeesh Pakkath,  Ayyiliath M. Sajith,  C. S. Ananda kumar,  Karickal R. Haridas,  M. Syed Ali Padusha, 
  • Pages: 2277-2283
  • First Published: 22 August 2018
A Highly Efficient Catalyst for the Suzuki-Miyaura Cross-Coupling Reaction of 5-(5-chloropyridin-3-yl)-3-methyl-1,3,4-oxadiazol-2(3H)-one

Reactions of N-alkenyl Thioureas with p-alkoxyphenyltellurium Trichlorides

Mykola Kut,  Maksym Fizer,  Mikhajlo Onysko,  Vasil Lendel, 
  • Pages: 2284-2290
  • First Published: 15 August 2018
Reactions of N-alkenyl Thioureas with p-alkoxyphenyltellurium Trichlorides

Preparation of Pyrido[2,3-b]indole Derivatives Using Silicates of Group 1 and 2 Metals

Setareh Sheikh,  Abbas Fazlinia, 
  • Pages: 2291-2296
  • First Published: 13 August 2018
Preparation of Pyrido[2,3-b]indole Derivatives Using Silicates of Group 1 and 2 Metals

Design, Synthesis and SAR Study of Novel Spiro [Pyrimido[5,4-b]Quinoline-10,5′-Pyrrolo[2,3-d]Pyrimidine] Derivatives as Promising Anticancer Agents

Asha V. Chate,  Sagar P. Kamdi,  Amruta N. Bhagat,  Chetan K. Jadhav,  Amol Nipte,  Aniket P. Sarkate,  Shailee V. Tiwari,  Charansingh H. Gill, 
  • Pages: 2297-2302
  • First Published: 13 August 2018
Design, Synthesis and SAR Study of Novel Spiro [Pyrimido[5,4-b]Quinoline-10,5′-Pyrrolo[2,3-d]Pyrimidine] Derivatives as Promising Anticancer Agents

Novel Pyrazolo[1,5-a]Pyrimidines and Pyrazolo[5,1-c][1,2,4]Triazines Incorporating Indole Moiety as a New Class of Antioxidant Agents

Ahmed El-Mekabaty,  Ahmed A. Fadda, 
  • Pages: 2303-2308
  • First Published: 15 August 2018
Novel Pyrazolo[1,5-a]Pyrimidines and Pyrazolo[5,1-c][1,2,4]Triazines Incorporating Indole Moiety as a New Class of Antioxidant Agents

Synthesis of Novel Structurally Diverse N-Mono- and N,N′-Disubstituted Benzimidazol-2-one Derivatives by the Alkylations of 1,3-Dihydro-2H-benzimidazol-2-one with Some Alkyl Halides under Transfer Catalysis Conditions

Taoufik Rohand,  Emmanuel Sopbué Fondjo, 
  • Pages: 2309-2314
  • First Published: 15 August 2018
Synthesis of Novel Structurally Diverse N-Mono- and N,N′-Disubstituted Benzimidazol-2-one Derivatives by the Alkylations of 1,3-Dihydro-2H-benzimidazol-2-one with Some Alkyl Halides under Transfer Catalysis Conditions

Studies on the Chemical Reactions of Some 3-Substituted-6,8-dimethylchromones with Nucleophilic Reagents

Magdy A. Ibrahim,  Al-Shimaa Badran,  Nasser M. El-Gohary,  Salsabeel H. Hashiem, 
  • Pages: 2315-2324
  • First Published: 22 August 2018
Studies on the Chemical Reactions of Some 3-Substituted-6,8-dimethylchromones with Nucleophilic Reagents

A Consecutive Condensation, Cyclization, and Dehydration for the Synthesis of Benzimidazopyrroloquinazolines Catalyzed by TsOH

Yi-Ping Wang,  Xue-Rong Ou,  Yue Wang,  Jian-Quan Liu,  Xiang-Shan Wang, 
  • Pages: 2325-2333
  • First Published: 17 August 2018
A Consecutive Condensation, Cyclization, and Dehydration for the Synthesis of Benzimidazopyrroloquinazolines Catalyzed by TsOH

Synthesis, Characterization, and Anticancer Activity (MCF-7) of Some Acetanilide-based Heterocycles

Ehab Abdel-Latif,  Eman M. Keshk,  Abdel-Galil M. Khalil,  Ali Saeed,  Heba M. Metwally, 
  • Pages: 2334-2341
  • First Published: 17 August 2018
Synthesis, Characterization, and Anticancer Activity (MCF-7) of Some Acetanilide-based Heterocycles

Synthesis of Novel Bis(thiazolylchromen-2-one) Derivatives Linked to Alkyl Spacer via Phenoxy Group

Mohamed Hosny,  Mostafa E. Salem,  Ahmed F. Darweesh,  Ahmed H. M. Elwahy, 
  • Pages: 2342-2348
  • First Published: 06 September 2018
Synthesis of Novel Bis(thiazolylchromen-2-one) Derivatives Linked to Alkyl Spacer via Phenoxy Group

Novel Bridgehead Thiadiazolopyrimidine Derivatives with Antimicrobial and Antitumor Activities

Mohammad E. Azab,  Salwa S. Abdel-Wahab,  Naglaa F. Mahmoud,  Galal A. Elsayed, 
  • Pages: 2349-2359
  • First Published: 17 August 2018
Novel Bridgehead Thiadiazolopyrimidine Derivatives with Antimicrobial and Antitumor Activities

Intramolecular Ring Transformation of Bis-oxadiazoles to Bis-thiadiazoles and Investigation of Their Anticancer Activities

Sobhi M. Gomha,  Zeinab A. Muhammad,  Ahmed A. M. El-Reedy, 
  • Pages: 2360-2367
  • First Published: 17 August 2018
Intramolecular Ring Transformation of Bis-oxadiazoles to Bis-thiadiazoles and Investigation of Their Anticancer Activities

Synthesis and Utility of α,β-Unsaturated Ketone Bearing Naphthalene and Benzofuran Rings in the Synthesis of Some N-heterocycles with Their Antiviral and Antitumor Activity Evaluation

Rasha S. Gouhar,  Ewies F. Ewies,  Mohamed F. El-Shehry,  Mohamed N. F. Shaheen,  El-Mahdy M. E. Ibrahim, 
  • Pages: 2368-2380
  • First Published: 31 August 2018
Synthesis and Utility of α,β-Unsaturated Ketone Bearing Naphthalene and Benzofuran Rings in the Synthesis of Some N-heterocycles with Their Antiviral and Antitumor Activity Evaluation

Grignard Reagents and Their N-analogues in the Synthesis of Tricyclic and Tetracyclic Cage-like Lactams

Igor V. Tkachenko,  Igor N. Tarabara,  Irina V. Omelchenko,  Vitalii A. Palchykov, 
  • Pages: 2381-2391
  • First Published: 31 August 2018
Grignard Reagents and Their N-analogues in the Synthesis of Tricyclic and Tetracyclic Cage-like Lactams

Molecular Modeling, Ionic Liquid Cu(II)-Catalyzed Synthesis of 9-(3-Fluoro-4-methoxyphenyl)-6-aryl-[1,2,4]triazolo[4,3-a][1,8] Naphthyridines under Microwave Irradiation and Their Antimicrobial Activity

Boda Sakram,  Kommakula Ashok,  Sirgamalla Rambabu,  Dharavath Ravi,  Adem Kurumanna,  Najlaa Khudhair Abbas, 
  • Pages: 2392-2399
  • First Published: 03 September 2018
Molecular Modeling, Ionic Liquid Cu(II)-Catalyzed Synthesis of 9-(3-Fluoro-4-methoxyphenyl)-6-aryl-[1,2,4]triazolo[4,3-a][1,8] Naphthyridines under Microwave Irradiation and Their Antimicrobial Activity

Synthesis, Antioxidant, and Antibacterial Activities of Some New 2-(3-fluorobenzyl)-1H-benzimidazole Derivatives

Hakan Bektas,  Canan Albay,  Bahar Bilgin Sökmen,  Sinem Aydın,  Emre Menteşe,  Gülbahar Aydın,  Dilem Şen, 
  • Pages: 2400-2407
  • First Published: 31 August 2018
Synthesis, Antioxidant, and Antibacterial Activities of Some New 2-(3-fluorobenzyl)-1H-benzimidazole Derivatives

Novel 4-Heteroaryl-antipyrines: Synthesis, Molecular Docking, and Evaluation as Potential Anti-breast Cancer Agents

Ziqi Tao,  Sobhi M. Gomha,  Mohamed G. Badrey,  Tamer T. El-Idreesy,  Taha M. A. Eldebss, 
  • Pages: 2408-2416
  • First Published: 30 August 2018
Novel 4-Heteroaryl-antipyrines: Synthesis, Molecular Docking, and Evaluation as Potential Anti-breast Cancer Agents

An Efficient Green Synthetic Approach to the Synthesis of 4H-Chromene Compounds under Solvent-free Conditions

Remon M. Zaki,  Saoud A. Metwally,  Yasser A. Elossaily,  Taher A. Gaber, 
  • Pages: 2417-2426
  • First Published: 30 August 2018
An Efficient Green Synthetic Approach to the Synthesis of 4H-Chromene Compounds under Solvent-free Conditions

Communications to the Editor

Interaction of Fused 1,2,4-Triazinone with Diborane/Oxidation: A New Route for the Synthesis of Partially Saturated and Aromatic Pyrazolo[5,1-c][1,2,4]triazines

Sergey M. Ivanov,  Anatoliy M. Shestopalov, 
  • Pages: 2427-2433
  • First Published: 08 August 2018
Interaction of Fused 1,2,4-Triazinone with Diborane/Oxidation: A New Route for the Synthesis of Partially Saturated and Aromatic Pyrazolo[5,1-c][1,2,4]triazines

Design, Synthesis, and Antibacterial Evaluation of Propylene-tethered 8-Methoxyl Ciprofloxacin-isatin Hybrids

Hua Guo, 
  • Pages: 2434-2440
  • First Published: 15 August 2018
Design, Synthesis, and Antibacterial Evaluation of Propylene-tethered 8-Methoxyl Ciprofloxacin-isatin Hybrids