• Issue

    Journal of Heterocyclic Chemistry: Volume 56, Issue 9

    2289-2694
    September 2019
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Issue Information

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Issue Information

  • Pages: 2289-2298
  • First Published: 13 September 2019

Reviews

Synthesis and Applications of 2-Substituted Imidazole and Its Derivatives: A Review

Drashti G. Daraji,  Neelam P. Prajapati,  Hitesh D. Patel, 
  • Pages: 2299-2317
  • First Published: 01 August 2019
Synthesis and Applications of 2-Substituted Imidazole and Its Derivatives: A Review

Diversified Synthetic Strategies for Pyrroloindoles: An Overview

Sundeep Kaur Manjal,  Shelly Pathania,  Rohit Bhatia,  Ramandeep Kaur,  Kapil Kumar,  Ravindra K. Rawal, 
  • Pages: 2318-2332
  • First Published: 16 August 2019
Diversified Synthetic Strategies for Pyrroloindoles: An Overview

Articles

An Unprecedented Synthesis of 3,3-Disubstituted Isochroman-1,4-diones Using Nitrones as Oxygen Atom Donors

Vidya Sathi,  Ani Deepthi,  Noble V. Thomas, 
  • Pages: 2333-2340
  • First Published: 17 July 2019
An Unprecedented Synthesis of 3,3-Disubstituted Isochroman-1,4-diones Using Nitrones as Oxygen Atom Donors

Ring Opening and Recyclization Reactions of 3-Nitrochromone with Some Nucleophilic Reagents

Magdy A. Ibrahim,  Youssef A. Alnamer, 
  • Pages: 2341-2346
  • First Published: 17 July 2019
Ring Opening and Recyclization Reactions of 3-Nitrochromone with Some Nucleophilic Reagents

Design, Regiospecific Green Synthesis, Chemical Computational Analysis, and Antimicrobial Evaluation of Novel Phthalazine Heterocycles

Sameh A. Rizk,  Salwa S. Abdelwahab,  Azza A. El-Badawy, 
  • Pages: 2347-2357
  • First Published: 30 July 2019
Design, Regiospecific Green Synthesis, Chemical Computational Analysis, and Antimicrobial Evaluation of Novel Phthalazine Heterocycles

Simple and Efficient Synthesis of Novel 3-Substituted 2-Thioxo-2,3-dihydro-1H-benzo[g]quinazolin-4-ones and Their Reactions with Alkyl Halides and α-Glycopyranosyl Bromides

Ahmed I. Khodair,  Mona A. Elsafi,  Siham A. Al-Issa, 
  • Pages: 2358-2368
  • First Published: 18 July 2019
Simple and Efficient Synthesis of Novel 3-Substituted 2-Thioxo-2,3-dihydro-1H-benzo[g]quinazolin-4-ones and Their Reactions with Alkyl Halides and α-Glycopyranosyl Bromides

Antimicrobial Properties of Some New Synthesized Benzothiazole Linked Carboxamide, Acetohydrazide, and Sulfonamide Systems

Ahmed A. Fadda,  Nanees N. Soliman,  Nesma M. Bayoumy, 
  • Pages: 2369-2378
  • First Published: 30 July 2019
Antimicrobial Properties of Some New Synthesized Benzothiazole Linked Carboxamide, Acetohydrazide, and Sulfonamide Systems

A Facile One-pot Synthesis and Anticancer Evaluation of Interesting Pyrazole and Pyrimidinthione via Heterocyclic Interconversion

Sameh A. Rizk,  Safa Shaban, 
  • Pages: 2379-2388
  • First Published: 17 July 2019
A Facile One-pot Synthesis and Anticancer Evaluation of Interesting Pyrazole and Pyrimidinthione via Heterocyclic Interconversion

Thermal Behavior Analysis of Two Synthesized Flavor Precursors of N-alkylpyrrole Derivatives

Lvye Ai,  Mengzhen Liu,  Xiaoming Ji,  Miao Lai,  Mingqin Zhao,  Tianbao Ren, 
  • Pages: 2389-2397
  • First Published: 16 July 2019
Thermal Behavior Analysis of Two Synthesized Flavor Precursors of N-alkylpyrrole Derivatives

ZnO Nanocatalyst Mediated Convergent Synthesis of Highly Substituted Imidazole and Imidazole-derived Bi-heterocyclic Scaffolds as Potential Antibacterial Agents

A. Jayashree,  B. Narayana,  Gauthama B. Uppine,  Vivek M. Ghate,  Shaila A. Lewis,  Bharathi Prakash,  Sarojini B. Kunhanna,  Madan S. Kumar, 
  • Pages: 2398-2410
  • First Published: 01 August 2019
ZnO Nanocatalyst Mediated Convergent Synthesis of Highly Substituted Imidazole and Imidazole-derived Bi-heterocyclic Scaffolds as Potential Antibacterial Agents

Synthesis, antimicrobial activity, and molecular docking study of formylnaphthalenyloxymethyl-triazolyl-N-phenylacetamides

Mahesh B. Muluk,  Sambhaji T. Dhumal,  Pramod S. Phatak,  Naziya N. M. A. Rehman,  Prashant P. Dixit,  Prafulla B. Choudhari,  Ramrao A. Mane,  Kishan P. Haval, 
  • Pages: 2411-2418
  • First Published: 17 July 2019
Synthesis, antimicrobial activity, and molecular docking study of formylnaphthalenyloxymethyl-triazolyl-N-phenylacetamides

Synthesis and Anticancer Evaluation of Some Novel Thiophene, Thieno[3,2-d]pyrimidine, Thieno[3,2-b]pyridine, and Thieno[3,2-e][1,4]oxazepine Derivatives Containing Benzothiazole Moiety

Aisha Y. Hassan,  Ebtehal M. Husseiny, 
  • Pages: 2419-2429
  • First Published: 18 July 2019
Synthesis and Anticancer Evaluation of Some Novel Thiophene, Thieno[3,2-d]pyrimidine, Thieno[3,2-b]pyridine, and Thieno[3,2-e][1,4]oxazepine Derivatives Containing Benzothiazole Moiety

Synthesis, Docking, and Pharmacological Evaluation of Derivatives of α-Aminoketones Appended to Sydnones as Potent Antitubercular and Antifungal Scaffolds

Atukuri Dorababu,  Ravindra R. Kamble,  Saba Kauser J. Shaikh,  Shilpa M. Somagond,  Praveen K. Bayannavar,  Shrinivas D. Joshi, 
  • Pages: 2430-2441
  • First Published: 31 July 2019
Synthesis, Docking, and Pharmacological Evaluation of Derivatives of α-Aminoketones Appended to Sydnones as Potent Antitubercular and Antifungal Scaffolds

Synthesis and In Vitro Urease Inhibition of Some Novel Benzimidazole-based Hydrazones

Emre Menteşe,  Bahar Bilgin Sökmen, 
  • Pages: 2442-2448
  • First Published: 30 July 2019
Synthesis and In Vitro Urease Inhibition of Some Novel Benzimidazole-based Hydrazones

Synthesis and Antibacterial Activity of Benzazolyl Azolyl Sulfamoyl Acetamides

Tankam Rajeswari,  Tamatam Rekha,  Guda Dinneswara Reddy,  Adivireddy Padmaja,  Venkatapuram Padmavathi, 
  • Pages: 2449-2459
  • First Published: 01 August 2019
Synthesis and Antibacterial Activity of Benzazolyl Azolyl Sulfamoyl Acetamides

Discovery of Novel Sulfonamide-Based 5-Arylidenerhodanines as Effective Carbonic Anhydrase (II) Inhibitors: Microwave-Assisted and Ultrasound-Assisted One-Pot Four-Component Synthesis, Molecular Docking, and Anti-CA II Screening Studies

Arif Mermer,  Neslihan Demirbas,  Ummuhan Cakmak,  Ahmet Colak,  Ahmet Demirbas,  Manikandan Alagumuthu,  Sivakumar Arumugam, 
  • Pages: 2460-2468
  • First Published: 30 July 2019
Discovery of Novel Sulfonamide-Based 5-Arylidenerhodanines as Effective Carbonic Anhydrase (II) Inhibitors: Microwave-Assisted and Ultrasound-Assisted One-Pot Four-Component Synthesis, Molecular Docking, and Anti-CA II Screening Studies

Et3N-Prompted Efficient Synthesis of Anthracenyl Pyrazolines and Their Cytotoxicity Evaluation against Cancer Cell Lines

Thechano Merry,  Prabhakar Maddela,  Kiran Devaraya,  Anand K. Kondapi,  Chullikkattil P. Pradeep, 
  • Pages: 2469-2478
  • First Published: 30 July 2019
Et3N-Prompted Efficient Synthesis of Anthracenyl Pyrazolines and Their Cytotoxicity Evaluation against Cancer Cell Lines

A Facile Synthesis of 2-Methyl-3-oxoindoline-2-carboxylates Utilizing Aza-Brook Rearrangement as a Crucial Step

Makoto Shimizu,  Haruna Katsurayama,  Isao Mizota,  Yusong Zhu, 
  • Pages: 2479-2486
  • First Published: 30 July 2019
A Facile Synthesis of 2-Methyl-3-oxoindoline-2-carboxylates Utilizing Aza-Brook Rearrangement as a Crucial Step

Efficient Synthesis and Antimicrobial Evaluation of New Azolopyrimidines-Bearing Pyrazole Moiety

Abdou O. Abdelhamid,  Sobhi M. Gomha,  Waleed A. M. A. El-Enany, 
  • Pages: 2487-2493
  • First Published: 29 July 2019
Efficient Synthesis and Antimicrobial Evaluation of New Azolopyrimidines-Bearing Pyrazole Moiety

Synthesis and Antifungal Activity of Substituted 2-Aryl Benzimidazoles Derivatives

Daye Huang,  Fang Qiu,  Zhigang Zhang,  Liqiao Shi,  Chunxia Cao,  Shaoyong Ke, 
  • Pages: 2494-2498
  • First Published: 30 July 2019
Synthesis and Antifungal Activity of Substituted 2-Aryl Benzimidazoles Derivatives

Synthesis and Characterization of Some BODIPY-based Substituted Salicylaldimine Schiff Bases

Nisha Kushwah,  Soumyaditya Mula,  Amey P. Wadawale,  Meenakshi Joshi,  Kedarnath Gotluru,  Mukesh Kumar,  Tapan K. Ghanty,  Sandip K. Nayak,  Vimal K. Jain, 
  • Pages: 2499-2507
  • First Published: 07 August 2019
Synthesis and Characterization of Some BODIPY-based Substituted Salicylaldimine Schiff Bases

Novel Approach for Rapid and Efficient Synthesis of 2-(3-(4-Aryl)-1-isonicotinoyl-4,5-dihydro-1H-pyrazol-4-yl)-3-phenylthiazolidin-4-one Derivatives and Screened Their Antimicrobial Activity

Meenu Beniwal,  Neelam Jain, 
  • Pages: 2508-2516
  • First Published: 14 August 2019
Novel Approach for Rapid and Efficient Synthesis of 2-(3-(4-Aryl)-1-isonicotinoyl-4,5-dihydro-1H-pyrazol-4-yl)-3-phenylthiazolidin-4-one Derivatives and Screened Their Antimicrobial Activity

One-pot Two-step Reaction for Synthesis of Poly-substituted Pyrano[3,2-c]pyridones and Spiro[indoline-3,4′-pyrano[3,2-c]pyridine]-2,5′(6′H)-diones in Water

Zhenhang Xu,  Yijun Du,  Songxiang Wang,  Zeru Wu,  Yuhao Lou,  Furen Zhang, 
  • Pages: 2517-2527
  • First Published: 05 August 2019
One-pot Two-step Reaction for Synthesis of Poly-substituted Pyrano[3,2-c]pyridones and Spiro[indoline-3,4′-pyrano[3,2-c]pyridine]-2,5′(6′H)-diones in Water

Synthesis and Antimicrobial and Antioxidant Activities of Sulfonamide Derivatives Containing Tetrazole and Oxadiazole Rings

Hamdi Özkan,  Bayram Demirci, 
  • Pages: 2528-2535
  • First Published: 11 August 2019
Synthesis and Antimicrobial and Antioxidant Activities of Sulfonamide Derivatives Containing Tetrazole and Oxadiazole Rings

Synthesis, Crystal Structure, Antifungal Activity, and Docking Study of Difluoromethyl Pyrazole Derivatives

Li Qiao,  Zhi-Wen Zhai,  Peng-Peng Cai,  Cheng-Xia Tan,  Jian-Quan Weng,  Liang Han,  Xing-Hai Liu,  Yong-Gang Zhang, 
  • Pages: 2536-2541
  • First Published: 06 August 2019
Synthesis, Crystal Structure, Antifungal Activity, and Docking Study of Difluoromethyl Pyrazole Derivatives

Synthesis, Density Functional Theory Band Structure Calculations, Optical, and Photoelectrical Characterizations of the Novel (9-Bromo-3-cyano-5-oxo-1,5-dihydro-2H-chromeno[4,3-b]pyridin-2-ylidene)propanedinitrile

Shimaa Abdel Halim,  Magdy A. Ibrahim, 
  • Pages: 2542-2554
  • First Published: 14 August 2019
Synthesis, Density Functional Theory Band Structure Calculations, Optical, and Photoelectrical Characterizations of the Novel (9-Bromo-3-cyano-5-oxo-1,5-dihydro-2H-chromeno[4,3-b]pyridin-2-ylidene)propanedinitrile

Novel Substituted Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives: Synthesis, Characterization, Molecular Docking Study, and Investigation of Their In Vitro Antifungal Activities

Mustafa Er,  Hakan Tahtaci,  Tuncay Karakurt,  Abdurrahman Onaran, 
  • Pages: 2555-2570
  • First Published: 13 August 2019
Novel Substituted Imidazo[2,1-b][1,3,4]Thiadiazole Derivatives: Synthesis, Characterization, Molecular Docking Study, and Investigation of Their In Vitro Antifungal Activities

Facile Synthesis, Antimicrobial Activity and Molecular Docking of Novel 2,4,5-Trisubstituted-1H-Imidazole–Triazole Hybrid Compounds

Sunil Chauhan,  Vikas Verma,  Devinder Kumar,  Ashwani Kumar, 
  • Pages: 2571-2579
  • First Published: 06 August 2019
Facile Synthesis, Antimicrobial Activity and Molecular Docking of Novel 2,4,5-Trisubstituted-1H-Imidazole–Triazole Hybrid Compounds

Design, Synthesis, and Pharmacological Assay of Novel Compounds Based on Pyridazine Moiety as Potential Antitumor Agents

Yasmeen M. Ali,  Mahmoud F. Ismail,  Fatma S. M. Abu El-Azm,  Magda I. Marzouk, 
  • Pages: 2580-2591
  • First Published: 12 August 2019
Design, Synthesis, and Pharmacological Assay of Novel Compounds Based on Pyridazine Moiety as Potential Antitumor Agents

Sequential Intramolecular Diels–Alder Reaction of 3-Heteroaryl-2-propenylamides of Ethenetricarboxylate

Hirotaka Sugiura,  Shoko Yamazaki,  Akiya Ogawa, 
  • Pages: 2592-2603
  • First Published: 18 August 2019
Sequential Intramolecular Diels–Alder Reaction of 3-Heteroaryl-2-propenylamides of Ethenetricarboxylate

Copper-Catalyzed N-Arylation of Polysubstituted Pyridines Synthesized by the Novel Reaction of N-Sulfonyl Ketenimine and Malononitrile-Trichloroacetonitrile Adduct

Manijeh Nematpour,  Hossein Fasihi Dastjerdi,  Sayyed Mohammad Ismaeil Mahboubi Rabbani,  Sayyed Abbas Tabatabai, 
  • Pages: 2604-2611
  • First Published: 14 August 2019
Copper-Catalyzed N-Arylation of Polysubstituted Pyridines Synthesized by the Novel Reaction of N-Sulfonyl Ketenimine and Malononitrile-Trichloroacetonitrile Adduct

Naked Eye Detection of Carbonate, Hydroxide, and Cyanide Ions with 1,4′-Diazaflavonium Bromides: A Simple Spectrophotometric Method for Cyanide Determination

Nuran Kahriman,  Serhat Gün,  Abidin Gümrükçüoğlu,  Nurettin Yaylı,  Ümmühan Ocak,  Miraç Ocak, 
  • Pages: 2612-2618
  • First Published: 18 August 2019
Naked Eye Detection of Carbonate, Hydroxide, and Cyanide Ions with 1,4′-Diazaflavonium Bromides: A Simple Spectrophotometric Method for Cyanide Determination

Functionalized Benzofurans via Microwave-Promoted Tandem Claisen-Rearrangement/5-endo-dig Cyclization

Christiane Schultze,  Bernd Schmidt, 
  • Pages: 2619-2629
  • First Published: 18 August 2019
Functionalized Benzofurans via Microwave-Promoted Tandem Claisen-Rearrangement/5-endo-dig Cyclization

A Convenient Synthesis of Bipyrido-Fused Coumarins and Their Biological Evaluation

Rakesh R. Giri,  Dinkar I. Brahmbhatt, 
  • Pages: 2630-2636
  • First Published: 16 August 2019
A Convenient Synthesis of Bipyrido-Fused Coumarins and Their Biological Evaluation

2-Cyano-N-(thiophen-2-yl)acetamide in Heterocyclic Synthesis: Synthesis and Antibacterial Screening of Novel Pyrido[1,2-a]thieno[3,2-e]pyrimidine-2-carboxylate Moieties

Amr M. Abdelmoniem,  Said A. S. Ghozlan,  Hassan M. Abdelwahab,  Ismail A. Abdelhamid, 
  • Pages: 2637-2643
  • First Published: 18 August 2019
2-Cyano-N-(thiophen-2-yl)acetamide in Heterocyclic Synthesis: Synthesis and Antibacterial Screening of Novel Pyrido[1,2-a]thieno[3,2-e]pyrimidine-2-carboxylate Moieties

Green Synthesis of Imidazole Derivatives via Fe3O4-MNPs as Reusable Catalyst

Faezeh Shafaei,  Shirin Sharafian, 
  • Pages: 2644-2650
  • First Published: 18 August 2019
Green Synthesis of Imidazole Derivatives via Fe3O4-MNPs as Reusable Catalyst

Highly Efficient [3 + 2] Cycloaddition: Click Synthesis of Novel 1H-indol-3-yl-benzo[d]imidazole Bis-triazoles

Mahesh Goud Bakkolla,  Ashok Kumar Taduri,  Rama Devi Bhoomireddy, 
  • Pages: 2651-2658
  • First Published: 14 August 2019
Highly Efficient [3 + 2] Cycloaddition: Click Synthesis of Novel 1H-indol-3-yl-benzo[d]imidazole Bis-triazoles

Notes

New Biphenyl-Based Bispyrazolines: Synthesis, Antimicrobial, and Docking Studies

Mohamad Yusuf,  Shehneela Nisa,  Kamaldeep Paul, 
  • Pages: 2659-2670
  • First Published: 05 August 2019
New Biphenyl-Based Bispyrazolines: Synthesis, Antimicrobial, and Docking Studies

Synthetic Study of Carthamin: Biomimetic Synthesis of Carthamin Model via Peroxidase-Catalyzed Oxidative Decarboxylation of Its Precursor Model

Takuo Sohtome,  Shingo Sato, 
  • Pages: 2671-2676
  • First Published: 29 July 2019
Synthetic Study of Carthamin: Biomimetic Synthesis of Carthamin Model via Peroxidase-Catalyzed Oxidative Decarboxylation of Its Precursor Model

Communications to the Editor

A Concise Stereoselective Synthesis of (R)-2-Benzylmorpholine and ML398 from (R)-(−)-2-Phenylglycinol

Saúl Torres,  Manuel Velasco,  José Ángel Gallegos-Rojas,  Sylvain Bernès,  María L. Orea,  Joel L. Terán,  Gabriela Huelgas,  Víctor Gómez-Calvario,  Jorge R. Juárez, 
  • Pages: 2677-2682
  • First Published: 13 August 2019
A Concise Stereoselective Synthesis of (R)-2-Benzylmorpholine and ML398 from (R)-(−)-2-Phenylglycinol

A Facile Synthesis of Raltegravir Potassium—An HIV Integrase Inhibitor

Kishore Karumanchi,  Gangadhara Bhima Shankar Nangi,  Subba Reddy Danda,  Ramadas Chavakula,  Raghu Babu Korupolu,  Kishore Babu Bonige, 
  • Pages: 2683-2690
  • First Published: 14 August 2019
A Facile Synthesis of Raltegravir Potassium—An HIV Integrase Inhibitor

Moxifloxacin/Gatifloxacin-1,2,3-triazole-isatin Hybrids with Hydrogen-Bond Donor and Their In Vitro Anticancer Activity

Rongxing Chen,  Hao Zhang,  Tianwei Ma,  Huarui Xue,  Zhong Miao,  Liyan Chen,  Xiangkui Shi, 
  • Pages: 2691-2694
  • First Published: 18 August 2019
Moxifloxacin/Gatifloxacin-1,2,3-triazole-isatin Hybrids with Hydrogen-Bond Donor and Their In Vitro Anticancer Activity