Isocyclic Compounds
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ChemInform Abstract: N-Cyclopropanation of Aromatic Amines.
First published: January 12, 1988
Abstract
The primary arylamines (Ia) and (Ib) and the secondary arylamines (Ic) are coupled with 1-bromo-1-ethoxycyclopropane (II) to produce the N-(1-ethoxycyclopropyl)arylamines (III).
ChemInform Abstract
The primary arylamines (Ia) and (Ib) and the secondary arylamines (Ic) are coupled with 1-bromo-1-ethoxycyclopropane (II) to produce the N-(1-ethoxycyclopropyl)arylamines (III). These compounds are reductively deethoxylated with sodium boranate in the presence of boron trifluoride etherate, yielding the N-arylcyclopropylamines (IV).
